Review of Recent Publications Featuring Binding Data Produced by Molecular Sensing’s Drug Discovery Services
Richard Isaacs, PhD
Wednesday, February 3, 2016
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Chapters
Introduction
Integral Membrane Protein Targets
Characterization of the direct interaction
Kv1.3 Binding Study
KCSA-Kv1.3 Chimera in Nanodiscs
SPR Binding for Peptide Ligands
BSI Binding for Peptides and Small Molecules
KCSA-Kv1.3 in Nanodiscs
Research Article
GPR39 Agonist Study
HTS Campaign for GPR39 Agonists
Functional Agonism Data
BSI Binding Data
Summary of Functional and BSI Assays
Summary
Thank You
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